Sfoglia per Autore
Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines
2010-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Sanna, M. L.; Gallinella, B.; Cirilli, R.
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
2011-01-01 Secci, D.; Carradori, Simone; Bolasco, A.; Chimenti, P.; Yáñez, M.; Ortuso, F.; Alcaro, S.
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
2011-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Lilli, D.; Rivanera, D.
Synthesis and biological evaluation of a new thiazole derivative, inducing histone hypoacetylation and apoptosis in human leukemia cells
2011-01-01 Carradori, Simone
Epigenetic modulation of PGC-1α activity by GCN5 inhibitors: WO2010007085
2011-01-01 Carradori, Simone; Secci, D.; Mai, A. .
The state of the art of pyrazole derivatives as monoamine oxidase inhibitors and antidepressant/anticonvulsant agents
2011-01-01 Secci, D.; Bolasco, A.; Chimenti, P.; Carradori, Simone
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines
2012-01-01 Secci, D.; Bolasco, A.; Carradori, Simone; D’Ascenzio, M.; Nescatelli, R.; Yáñez, M.
Conventional and microwave-assisted synthesis of benzimidazole derivatives and their in vitro inhibition of human cyclooxygenase
2012-01-01 Secci, D.; Bolasco, A.; D’Ascenzio, M.; della Sala, F.; Yáñez, M.; Carradori, Simone
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
2012-01-01 Secci, D.; Bizzarri, B.; Bolasco, A.; Carradori, Simone; D'Ascenzio, M.; Rivanera, D.; Mari, E.; Polletta, L.; Zicari, A.
3-Methylcyclohexanone thiosemicarbazone: determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes
2012-01-01 Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, S.; Pierini, M.; Secci, D.
Current and emerging strategies in bladder cancer
2012-01-01 Carradori, Simone; Cristini, C.; Secci, D.; Gulia, C.; Gentile, V.; Di Pierro, G. B.
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
2012-01-01 Secci, D.; Carradori, Simone; Bolasco, A.; Bizzarri, B.; D’Ascenzio, M.; Maccioni, E.
CPTH6, a thiazole-derivative, induces histone hypoacetylation and apoptosis in human leukemia cells
2012-01-01 Trisciuoglio, D.; Ragazzoni, Y.; Pelosi, A.; Desideri, M.; Carradori, Simone; Gabellini, C.; Maresca, G.; Nescatelli, R.; Secci, D.; Bolasco, A.; Bizzarri, B.; Cavaliere, C.; D'Agnano, I.; Filetici, P.; Ricci Vitiani, L.; Rizzo, M. G.; Del Bufalo, D.
Thiazolidinone scaffold: a new pharmacophore for anti-Toxoplasma gondii agents
2012-01-01 Carradori, Simone; De Monte, C.; Bizzari, B.; Secci, D.; Jones Brando, L.
Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives
2012-01-01 Carradori, Simone; Secci, D.; Bolasco, A.; De Monte, C.; Yáñez, M.
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
2012-01-01 Carradori, Simone; Secci, D.; Bolasco, A.; Chimenti, P.; D'Ascenzio, M.
Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII - A new scaffold for designing isoform-selective inhibitors
2013-01-01 Carradori, Simone; De Monte, C.; D’Ascenzio, M.; Secci, D.; Celik, G.; Ceruso, M.; Vullo, D.; Scozzafava, A.; Supuran, C. T.
Muscle-invasive and metastatic bladder cancer: current and emerging therapies
2013-01-01 Pietro, Grande; Carradori, Simone; Cristiano, Cristini; Daniela, Secci; Caterina, Gulia; Vincenzo, Gentile; Giovanni Di, Pierro
Synthesis and selective human MAO-B inhibition of heterocyclic hybrids based on hydrazine and thiazole scaffolds
2013-01-01 Carradori, Simone; D’Ascenzio, M.; De Monte, C.; Secci, D.; Yáñez, M.
Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors
2013-01-01 Chimenti, P.; Petzer, A.; Carradori, Simone; D’Ascenzio, M.; Silvestri, R.; Alcaro, S.; Ortuso, F.; Petzer, J. P.; Secci, D.
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