Sfoglia per Autore
Discovery of 7-aminophenanthridin-6-one as a new scaffold for matrix metalloproteinase inhibitors with multitarget neuroprotective activity
2021-01-01 Rocchi, Damiano; Blázquez-Barbadillo, Cristina; Agamennone, Mariangela; Laghezza, Antonio; Tortorella, Paolo; Vicente-Zurdo, David; Rosales-Conrado, Noelia; Moyano, Paula; Del Pino, Javier; F González, Juan; Carlos Menéndez, J
(2-Aminobenzothiazole)-Methyl-1,1-bisphosphonic acids: Targeting matrix metalloproteinase 13 inhibition to the bone
2021-01-01 Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Loiodice, F.; Tortorella, P.
Development of CDK4/6 Inhibitors: A Five Years Update
2021-01-01 Ammazzalorso, Alessandra; Agamennone, Mariangela; De Filippis, Barbara; Fantacuzzi, Marialuigia
Discovery of a novel tetrapeptide against influenza a virus: Rational design, synthesis, bioactivity evaluation and computational studies
2021-01-01 Scala, Maria Carmina; Agamennone, Mariangela; Pietrantoni, Agostina; Di Sarno, Veronica; Bertamino, Alessia; Superti, Fabiana; Campiglia, Pietro; Sala, Marina
Hampering the early aggregation of PrP-E200K protein by charge-based inhibitors: a computational study
2021-01-01 Agamennone, M.; Storchi, L.; Marrone, A.; Paciotti, R.
Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure-Activity Relationship Studies and Target Prediction Analysis
2022-01-01 Amoroso, R; De Lellis, L; Florio, R; Moreno, N; Agamennone, M; De Filippis, B; Giampietro, L; Maccallini, C; Fernández, I; Recio, R; Cama, A; Fantacuzzi, M; Ammazzalorso, A.
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?
2022-01-01 Carradori, S.; Fantacuzzi, M.; Ammazzalorso, A.; Angeli, A.; De Filippis, B.; Galati, S.; Petzer, A.; Petzer, J. P.; Poli, G.; Tuccinardi, T.; Agamennone, M.; Supuran, C. T.
Antiviral Peptides as Anti-Influenza Agents
2022-01-01 Agamennone, Mariangela; Fantacuzzi, Marialuigia; Vivenzio, Giovanni; Scala, Maria Carmina; Campiglia, Pietro; Superti, Fabiana; Sala, Marina
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies
2022-01-01 Agamennone, M.; Fantacuzzi, M.; Carradori, S.; Petzer, A.; Petzer, J. P.; Angeli, A.; Supuran, C. T.; Luisi, G.
Het(aryl)isatin to het(aryl)aminoindoline scaffold hopping: A route to selective inhibitors of matrix metalloproteinases
2022-01-01 Ivanov, Vladimir N.; Agamennone, Mariangela; Iusupov, Ildar R.; Laghezza, Antonio; Novoselov, Anton M.; Manasova, Ekaterina V.; Altieri, Andrea; Tortorella, Paolo; Shtil, Alexander A.; Kurkin, Alexander V.
Broad-Spectrum Activity of Small Molecules Acting against Influenza a Virus: Biological and Computational Studies
2022-01-01 Agamennone, M.; Superti, F.
Erlotinib-containing benzenesulfonamides as anti-Helicobacter pylori agents through carbonic anhydrase inhibition
2023-01-01 Benito, G.; D'Agostino, I.; Carradori, S.; Fantacuzzi, M.; Agamennone, M.; Puca, V.; Grande, R.; Capasso, C.; Carta, F.; Supuran, C. T.
Identification of Anti-Influenza A Compounds Inhibiting the Viral Non-Structural Protein 1 (NS1) Using a Type I Interferon-Driven Screening Strategy
2023-01-01 Marsili, Giulia; Acchioni, Chiara; Remoli, Anna Lisa; Amatore, Donatella; Sgarbanti, Rossella; De Angelis, Marta; Orsatti, Roberto; Acchioni, Marta; Astolfi, Andrea; Iraci, Nunzio; Puzelli, Simona; Facchini, Marzia; Perrotti, Edvige; Cecchetti, Violetta; Sabatini, Stefano; Superti, Fabiana; Agamennone, Mariangela; Barreca, Maria Letizia; Hiscott, John; Nencioni, Lucia; Sgarbanti, Marco
Rational Design of Novel Peptidomimetics against Influenza A Virus: Biological and Computational Studies
2023-01-01 Scala, Maria Carmina; Marchetti, Magda; Superti, Fabiana; Agamennone, Mariangela; Campiglia, Pietro; Sala, Marina
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships
2023-01-01 Fantacuzzi, M.; D'Agostino, I.; Carradori, S.; Liguori, F.; Carta, F.; Agamennone, M.; Angeli, A.; Sannio, F.; Docquier, J. -D.; Capasso, C.; Supuran, C. T.
A Comprehensive Computational Insight into the PD-L1 Binding to PD-1 and Small Molecules
2024-01-01 Fantacuzzi, Marialuigia; Paciotti, Roberto; Agamennone, Mariangela
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Discovery of 7-aminophenanthridin-6-one as a new scaffold for matrix metalloproteinase inhibitors with multitarget neuroprotective activity | 2021 | Rocchi, Damiano; Blázquez-Barbadillo, Cristina; Agamennone, Mariangela; Laghezza, Antonio; Tortorella, Paolo; Vicente-Zurdo, David; Rosales-Conrado, Noelia; Moyano, Paula; Del Pino, Javier; F González, Juan; Carlos Menéndez, J | |
(2-Aminobenzothiazole)-Methyl-1,1-bisphosphonic acids: Targeting matrix metalloproteinase 13 inhibition to the bone | 2021 | Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Loiodice, F.; Tortorella, P. | |
Development of CDK4/6 Inhibitors: A Five Years Update | 2021 | Ammazzalorso, Alessandra; Agamennone, Mariangela; De Filippis, Barbara; Fantacuzzi, Marialuigia | |
Discovery of a novel tetrapeptide against influenza a virus: Rational design, synthesis, bioactivity evaluation and computational studies | 2021 | Scala, Maria Carmina; Agamennone, Mariangela; Pietrantoni, Agostina; Di Sarno, Veronica; Bertamino, Alessia; Superti, Fabiana; Campiglia, Pietro; Sala, Marina | |
Hampering the early aggregation of PrP-E200K protein by charge-based inhibitors: a computational study | 2021 | Agamennone, M.; Storchi, L.; Marrone, A.; Paciotti, R. | |
Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure-Activity Relationship Studies and Target Prediction Analysis | 2022 | Amoroso, R; De Lellis, L; Florio, R; Moreno, N; Agamennone, M; De Filippis, B; Giampietro, L; Maccallini, C; Fernández, I; Recio, R; Cama, A; Fantacuzzi, M; Ammazzalorso, A. | |
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases? | 2022 | Carradori, S.; Fantacuzzi, M.; Ammazzalorso, A.; Angeli, A.; De Filippis, B.; Galati, S.; Petzer, A.; Petzer, J. P.; Poli, G.; Tuccinardi, T.; Agamennone, M.; Supuran, C. T. | |
Antiviral Peptides as Anti-Influenza Agents | 2022 | Agamennone, Mariangela; Fantacuzzi, Marialuigia; Vivenzio, Giovanni; Scala, Maria Carmina; Campiglia, Pietro; Superti, Fabiana; Sala, Marina | |
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies | 2022 | Agamennone, M.; Fantacuzzi, M.; Carradori, S.; Petzer, A.; Petzer, J. P.; Angeli, A.; Supuran, C. T.; Luisi, G. | |
Het(aryl)isatin to het(aryl)aminoindoline scaffold hopping: A route to selective inhibitors of matrix metalloproteinases | 2022 | Ivanov, Vladimir N.; Agamennone, Mariangela; Iusupov, Ildar R.; Laghezza, Antonio; Novoselov, Anton M.; Manasova, Ekaterina V.; Altieri, Andrea; Tortorella, Paolo; Shtil, Alexander A.; Kurkin, Alexander V. | |
Broad-Spectrum Activity of Small Molecules Acting against Influenza a Virus: Biological and Computational Studies | 2022 | Agamennone, M.; Superti, F. | |
Erlotinib-containing benzenesulfonamides as anti-Helicobacter pylori agents through carbonic anhydrase inhibition | 2023 | Benito, G.; D'Agostino, I.; Carradori, S.; Fantacuzzi, M.; Agamennone, M.; Puca, V.; Grande, R.; Capasso, C.; Carta, F.; Supuran, C. T. | |
Identification of Anti-Influenza A Compounds Inhibiting the Viral Non-Structural Protein 1 (NS1) Using a Type I Interferon-Driven Screening Strategy | 2023 | Marsili, Giulia; Acchioni, Chiara; Remoli, Anna Lisa; Amatore, Donatella; Sgarbanti, Rossella; De Angelis, Marta; Orsatti, Roberto; Acchioni, Marta; Astolfi, Andrea; Iraci, Nunzio; Puzelli, Simona; Facchini, Marzia; Perrotti, Edvige; Cecchetti, Violetta; Sabatini, Stefano; Superti, Fabiana; Agamennone, Mariangela; Barreca, Maria Letizia; Hiscott, John; Nencioni, Lucia; Sgarbanti, Marco | |
Rational Design of Novel Peptidomimetics against Influenza A Virus: Biological and Computational Studies | 2023 | Scala, Maria Carmina; Marchetti, Magda; Superti, Fabiana; Agamennone, Mariangela; Campiglia, Pietro; Sala, Marina | |
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships | 2023 | Fantacuzzi, M.; D'Agostino, I.; Carradori, S.; Liguori, F.; Carta, F.; Agamennone, M.; Angeli, A.; Sannio, F.; Docquier, J. -D.; Capasso, C.; Supuran, C. T. | |
A Comprehensive Computational Insight into the PD-L1 Binding to PD-1 and Small Molecules | 2024 | Fantacuzzi, Marialuigia; Paciotti, Roberto; Agamennone, Mariangela |
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