Sfoglia per Titolo
Synthesis and biological characterization of 3-(imidazol-1-ylmethyl)piperidine sulfonamides as aromatase inhibitors
2016-01-01 DI MATTEO, Mauro; Ammazzalorso, Alessandra; Andreoli, Federico; Caffa, Irene; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Maccallini, Cristina; Nencioni, Alessio; Parenti, Marco Daniele; Soncini, Debora; Rio, Alberto Del; Amoroso, Rosa
synthesis and biological evaluation as anti-Parkinson agent of an analogue of Glutathione-L-Dopa containing methionine in place of the cysteinil residue
2009-01-01 Cacciatore, Ivana; Cornacchia, Catia; Mollica, Adriano; Feliciani, Federica; DI STEFANO, Antonio; Sozio, Piera; Iannitelli, Antonio; Cerasa, LAURA SERAFINA; Pinnen, Francesco Enrico
Synthesis and Biological Evaluation of 2-Heteroarylthioalkanoic Acid Analogues of Clofibric Acid as Peroxisome Proliferator-Activated Receptor alfa Agonists
2009-01-01 Giampietro, Letizia; Ammazzalorso, Alessandra; Giancristofaro, Antonella; Lannutti, Fabio; Bettoni, Giancarlo; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Maccallini, Cristina; Petruzzelli, Michele; Morgano, Annalisa; Moschetta, Antonio; Amoroso, Rosa
Synthesis and biological evaluation of a new thiazole derivative, inducing histone hypoacetylation and apoptosis in human leukemia cells
2011-01-01 Carradori, Simone
Synthesis and biological evaluation of a novel pyroglutamil-modified TRH analogue
2002-01-01 Brunetti, Luigi; Cacciatore, Ivana; DI STEFANO, Antonio; Dupre', S; Giorgi, A; Luisi, Grazia; Michelotto, B; Orlando, Giustino; Pinnen, Francesco Enrico; Recinella, Lucia; Sozio, Piera; Spirito, A.
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
2017-01-01 Carradori, Simone; Secci, D.; Bizzarri, B.; Chimenti, P.; De Monte, C.; Guglielmi, P.; Campestre, Cristina; Rivanera, D.; Bordón, C.; Jones Brando, L.
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation
2020-01-01 Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Marcantonio, M. C. D.; Haloci, E.; Grande, R.; Mincione, G.
Synthesis and Biological Evaluation of GABA Derivatives Able to Cross the Blood-Brain Barrier in Rats
2003-01-01 Carelli, V.; Liberatore, F.; Scipione, L. GIORGIONI G.; DI STEFANO, Antonio; Impicciatore, M.; Ballabeni, V.; Calcina, F.; Magnanini, F.; Barocelli, E.
Synthesis and biological evaluation of gemfibrozil chiral analogs as potential PPARa agonists
2011-01-01 DE FILIPPIS, Barbara; Giampietro, Letizia; Giancristofaro, Antonella; Ammazzalorso, Alessandra; Fantacuzzi, Marialuigia; Maccallini, Cristina; Petruzzelli, Michele; Amoroso, Rosa
Synthesis and Biological Evaluation of Halogenated E-Stilbenols as Promising Antiaging Agents
2020-01-01 DI FILIPPO, ESTER SARA; Giampietro, Letizia; DE FILIPPIS, Barbara; Balaha, MARWA FATHY HASAN; Ferrone, Vincenzo; Locatelli, Marcello; Pietrangelo, Tiziana; Tartaglia, Angela; Amoroso, Rosa; Fulle, Stefania
Synthesis and biological evaluation of new 3(2H)-pyridazinone derivatives as non-toxic anti-proliferative compounds against human colon carcinoma HCT116 cells
2020-01-01 Ozdemir, Z.; Utku, S.; Mathew, B.; Carradori, S.; Orlando, G.; Di Simone, S.; Alagoz, M. A.; Ozcelik, A. B.; Uysal, M.; Ferrante, C.
Synthesis and biological evaluation of new acetamidines as selective inhibitors of Nitric Oxide Synthases
2013-01-01 DI MATTEO, Mauro; Maccallini, Cristina; Ammazzalorso, Alessandra; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Pandolfi, Assunta; Re, Nazzareno; Amoroso, Rosa
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues
2012-01-01 Mollica, Adriano; Feliciani, Federica; Stefanucci, Azzurra; Costante, Roberto; Gino, Lucente; Pinnen, Francesco Enrico; D., Notaristefano; S., Spisani
Synthesis and biological evaluation of new biphalin analogues with non-hydrazine linkers
2005-01-01 Mollica, Adriano; Davis, P; Ma, S. W.; Lai, J; Porreca, F; Hruby, V. J.
Synthesis and biological evaluation of new linear and cyclic Biphalin analogues
2005-01-01 Mollica, Adriano
Synthesis and biological evaluation of new matrix metalloproteinases inhibitors
2002-01-01 Agamennone, Mariangela; Tortorella, Paolo; Lucci, Sabrina; Campestre, Cristina; M., Crucianelli; A., Aramini; R., Ragno; F., Mazza; Gallina, Carlo
Synthesis and biological evaluation of new Matrix Metalloproteinases Inhibitors.
2003-01-01 Campestre, Cristina; Preziuso, Serena; Agamennone, Mariangela; Tortorella, Paolo; Gallina, Carlo
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
2011-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Lilli, D.; Rivanera, D.
Synthesis and biological evaluation of novel acetamidines as nitric oxide inhibitors
2010-01-01 Fantacuzzi, Marialuigia; Maccallini, Cristina; Patruno, Antonia; Masella, Simona; Di Tullio, M.; Tricca, M. L.; Amoroso, Rosa
Synthesis and biological evaluation of novel analogues of Gly-l-Pro-l-Glu (GPE) as neuroprotective agents
2019-01-01 Marinelli, Lisa; Fornasari, Erika; Di Stefano, Antonio; Turkez, Hasan; Genovese, Salvatore; Epifano, Francesco; Di Biase, Giuseppe; Costantini, Erica; D'Angelo, Chiara; Reale, Marcella; Cacciatore, Ivana
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and biological characterization of 3-(imidazol-1-ylmethyl)piperidine sulfonamides as aromatase inhibitors | 2016 | DI MATTEO, Mauro; Ammazzalorso, Alessandra; Andreoli, Federico; Caffa, Irene; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Maccallini, Cristina; Nencioni, Alessio; Parenti, Marco Daniele; Soncini, Debora; Rio, Alberto Del; Amoroso, Rosa | |
synthesis and biological evaluation as anti-Parkinson agent of an analogue of Glutathione-L-Dopa containing methionine in place of the cysteinil residue | 2009 | Cacciatore, Ivana; Cornacchia, Catia; Mollica, Adriano; Feliciani, Federica; DI STEFANO, Antonio; Sozio, Piera; Iannitelli, Antonio; Cerasa, LAURA SERAFINA; Pinnen, Francesco Enrico | |
Synthesis and Biological Evaluation of 2-Heteroarylthioalkanoic Acid Analogues of Clofibric Acid as Peroxisome Proliferator-Activated Receptor alfa Agonists | 2009 | Giampietro, Letizia; Ammazzalorso, Alessandra; Giancristofaro, Antonella; Lannutti, Fabio; Bettoni, Giancarlo; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Maccallini, Cristina; Petruzzelli, Michele; Morgano, Annalisa; Moschetta, Antonio; Amoroso, Rosa | |
Synthesis and biological evaluation of a new thiazole derivative, inducing histone hypoacetylation and apoptosis in human leukemia cells | 2011 | Carradori, Simone | |
Synthesis and biological evaluation of a novel pyroglutamil-modified TRH analogue | 2002 | Brunetti, Luigi; Cacciatore, Ivana; DI STEFANO, Antonio; Dupre', S; Giorgi, A; Luisi, Grazia; Michelotto, B; Orlando, Giustino; Pinnen, Francesco Enrico; Recinella, Lucia; Sozio, Piera; Spirito, A. | |
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives | 2017 | Carradori, Simone; Secci, D.; Bizzarri, B.; Chimenti, P.; De Monte, C.; Guglielmi, P.; Campestre, Cristina; Rivanera, D.; Bordón, C.; Jones Brando, L. | |
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation | 2020 | Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Marcantonio, M. C. D.; Haloci, E.; Grande, R.; Mincione, G. | |
Synthesis and Biological Evaluation of GABA Derivatives Able to Cross the Blood-Brain Barrier in Rats | 2003 | Carelli, V.; Liberatore, F.; Scipione, L. GIORGIONI G.; DI STEFANO, Antonio; Impicciatore, M.; Ballabeni, V.; Calcina, F.; Magnanini, F.; Barocelli, E. | |
Synthesis and biological evaluation of gemfibrozil chiral analogs as potential PPARa agonists | 2011 | DE FILIPPIS, Barbara; Giampietro, Letizia; Giancristofaro, Antonella; Ammazzalorso, Alessandra; Fantacuzzi, Marialuigia; Maccallini, Cristina; Petruzzelli, Michele; Amoroso, Rosa | |
Synthesis and Biological Evaluation of Halogenated E-Stilbenols as Promising Antiaging Agents | 2020 | DI FILIPPO, ESTER SARA; Giampietro, Letizia; DE FILIPPIS, Barbara; Balaha, MARWA FATHY HASAN; Ferrone, Vincenzo; Locatelli, Marcello; Pietrangelo, Tiziana; Tartaglia, Angela; Amoroso, Rosa; Fulle, Stefania | |
Synthesis and biological evaluation of new 3(2H)-pyridazinone derivatives as non-toxic anti-proliferative compounds against human colon carcinoma HCT116 cells | 2020 | Ozdemir, Z.; Utku, S.; Mathew, B.; Carradori, S.; Orlando, G.; Di Simone, S.; Alagoz, M. A.; Ozcelik, A. B.; Uysal, M.; Ferrante, C. | |
Synthesis and biological evaluation of new acetamidines as selective inhibitors of Nitric Oxide Synthases | 2013 | DI MATTEO, Mauro; Maccallini, Cristina; Ammazzalorso, Alessandra; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Pandolfi, Assunta; Re, Nazzareno; Amoroso, Rosa | |
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues | 2012 | Mollica, Adriano; Feliciani, Federica; Stefanucci, Azzurra; Costante, Roberto; Gino, Lucente; Pinnen, Francesco Enrico; D., Notaristefano; S., Spisani | |
Synthesis and biological evaluation of new biphalin analogues with non-hydrazine linkers | 2005 | Mollica, Adriano; Davis, P; Ma, S. W.; Lai, J; Porreca, F; Hruby, V. J. | |
Synthesis and biological evaluation of new linear and cyclic Biphalin analogues | 2005 | Mollica, Adriano | |
Synthesis and biological evaluation of new matrix metalloproteinases inhibitors | 2002 | Agamennone, Mariangela; Tortorella, Paolo; Lucci, Sabrina; Campestre, Cristina; M., Crucianelli; A., Aramini; R., Ragno; F., Mazza; Gallina, Carlo | |
Synthesis and biological evaluation of new Matrix Metalloproteinases Inhibitors. | 2003 | Campestre, Cristina; Preziuso, Serena; Agamennone, Mariangela; Tortorella, Paolo; Gallina, Carlo | |
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents | 2011 | Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Lilli, D.; Rivanera, D. | |
Synthesis and biological evaluation of novel acetamidines as nitric oxide inhibitors | 2010 | Fantacuzzi, Marialuigia; Maccallini, Cristina; Patruno, Antonia; Masella, Simona; Di Tullio, M.; Tricca, M. L.; Amoroso, Rosa | |
Synthesis and biological evaluation of novel analogues of Gly-l-Pro-l-Glu (GPE) as neuroprotective agents | 2019 | Marinelli, Lisa; Fornasari, Erika; Di Stefano, Antonio; Turkez, Hasan; Genovese, Salvatore; Epifano, Francesco; Di Biase, Giuseppe; Costantini, Erica; D'Angelo, Chiara; Reale, Marcella; Cacciatore, Ivana |
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