Sfoglia per Titolo
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
2017-01-01 Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; De Monte, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela
Synthesis, biological evaluation, and docking study of indole aryl sulfonamides as aromatase inhibitors
2020-01-01 Fantacuzzi, M.; De Filippis, B.; Gallorini, M.; Ammazzalorso, A.; Giampietro, L.; Maccallini, C.; Aturki, Z.; Donati, E.; Ibrahim, R. S.; Shawky, E.; Cataldi, A.; Amoroso, R.
Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity.
2008-01-01 Anzini, M; Rovini, M; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Giordani, A; Makovec, F; Anzellotti, P; Patrignani, Paola; Biava, M.
Synthesis, biological evaluation, and molecular modeling of oleuropein and its semisynthetic derivatives as cyclooxygenase inhibitors
2009-01-01 Procopio, A; Alcaro, S; Nardi, M; Oliverio, M; Ortuso, F; Sacchetta, Paolo; Pieragostino, Damiana; Sindona, G.
“Synthesis, characterisation and application of a novel thiophene-based polymer”
2005-01-01 Cheylan, S; Fraleoni Morgera, A; Puigdollers, J; Voz, C; Alcubilla, R; Setti, L; Badenes, G
Synthesis, characterization and evaluation of gemfibrozil-stilbene hybrid as antioxidant agent
2018-01-01 Amoroso, Rosa; Leporini, Lidia; Cacciatore, Ivana; Marinelli, Lisa; Ammazzalorso, Alessandra; Bruno, Isabella; De Filippis, Barbara; Fantacuzzi, Marialuigia; Maccallini, Cristina; Menghini, Luigi; Di Stefano, Antonio; Giampietro, Letizia
Synthesis, characterization and optical properties of a regioregular and soluble poly [3-(10-hydroxydecyl)-2,5-thienylene]
2003-01-01 Lanzi, Massimiliano; Costa-Bizzarri, Paolo; Della-Casa, Carlo; FRALEONI MORGERA, Alessandro; Paganin, Luisa
Synthesis, characterization, and antibacterial activity of chitosan-chelated silver nanoparticles.
2024-01-01 Ge, J; Li, M; Fan, J; Celia, C; Xie, Y; Chang, Q; Deng, X.
Synthesis, characterization, and computational study of aggregates from amphiphilic calix[6]arenes. Effect of encapsulation on degradation kinetics of curcumin
2022-01-01 Moffa, S.; Aschi, M.; Bazzoni, M.; Cester Bonati, F.; Secchi, A.; Bruni, P.; Di Profio, P.; Fontana, A.; Pilato, S.; Siani, G.
Synthesis, Characterization, and DNA Binding Profile of a Macrocyclic β-Sheet Analogue of ARC Protein
2015-01-01 Stefanucci, Azzurra; Mosquera, Jesús; Vázquez, Eugènio; Mascareñas, José L.; Novellino, Ettore; Mollica, Adriano
Synthesis, crystal structure and crystal-chemistry of ferri-clinoholmquistite, Li2Mg3Fe3+2Si8O22(OH)2.
2004-01-01 Iezzi, Gianluca; Camara, F.; DELLA VENTURA, G.; Oberti, R.; Pedrazzi, G.; Robert, J. L.
Synthesis, crystal structure, and magnetic properties of a ferrimagnetic layered compound [NEt(4)][Mn(5-Cl-salen)](2)[Fe(CN)(6)] (NEt(4) equals tetraethylammonium, 5-Cl-salen equals N,N'-ethylenebis((5-chlorosalicylidene)aminato))
1997-01-01 H., Miyasaka; N., Matsumoto; Re, Nazzareno; E., Gallo; C., Floriani
Synthesis, cytotoxicity and anti−proliferative activity against ags cells of new 3(2h)−pyridazinone derivatives endowed with a piperazinyl linker
2021-01-01 Alagoz, M. A.; Ozdemir, Z.; Uysal, M.; Carradori, S.; Gallorini, M.; Ricci, A.; Zara, S.; Mathew, B.
Synthesis, in vitro evaluation, and molecular modelling investigation of benzenesulfonimide Peroxisome Proliferator-Activated Receptors α antagonists
2016-01-01 Ammazzalorso, Alessandra; Carrieri, Antonio; Verginelli, Fabio; Bruno, Isabella; Carbonara, Giuseppe; D'Angelo, Alessandra; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Florio, Rosalba; Fracchiolla, Giuseppe; Giampietro, Letizia; Giancristofaro, Antonella; Maccallini, Cristina; Cama, Alessandro; Amoroso, Rosa
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents.
2008-01-01 Biava, M; Porretta, Gc; Poce, G; Supino, S; Manetti, F; Forli, S; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Giordani, A; Anzellotti, P; Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Anzini, M; Patrignani, Paola
Synthesis, magnetic properties, and incomplete double-cubane structure of Manganese(III)-metal(II) complexes [Mn(MeOH)L(OH)M(bpy)](2) (M = Zn, Cu, Ni, and Mn; H4L = 1,2-bis(2-hydroxybenzamido)benzene; bpy = 2,2 '-bipyridine)
1998-01-01 Y., Sunatsuki; H., Shimada; T., Matsuo; M., Nakamura; F., Kai; N., Matsumoto; Re, Nazzareno
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N’-bis[2-oxo-2H-benzopyran]-3-carboxamides
2006-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Befani, O.; Turini, P.; Alcaro, S.; Ortuso, F.
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins
2009-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Bizzarri, B.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Ortuso, F.; Alcaro, S.
Synthesis, pharmacological characterization, and docking analysis of a novel family of diarylisoxazoles as highly selective cyclooxygenase-1 (COX-1) inhibitors.
2013-01-01 Vitale, P; Tacconelli, Stefania; Perrone, Mg; Malerba, P; Simone, L; Scilimati, A; Lavecchia, A; Dovizio, Melania; Marcantoni, Emanuela; Bruno, Annalisa; Patrignani, Paola
Synthesis, Resolution, and Preliminary Evaluation of trans-2-amino-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes and Related Derivatives as Dopamine Receptors ligands
1996-01-01 Claudi, F; Cingolani, G. M.; DI STEFANO, Antonio; Giorgioni, G; Amenta, F; Barili, P; Ferrari, F; Giuliani, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity | 2017 | Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; De Monte, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela | |
Synthesis, biological evaluation, and docking study of indole aryl sulfonamides as aromatase inhibitors | 2020 | Fantacuzzi, M.; De Filippis, B.; Gallorini, M.; Ammazzalorso, A.; Giampietro, L.; Maccallini, C.; Aturki, Z.; Donati, E.; Ibrahim, R. S.; Shawky, E.; Cataldi, A.; Amoroso, R. | |
Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity. | 2008 | Anzini, M; Rovini, M; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Giordani, A; Makovec, F; Anzellotti, P; Patrignani, Paola; Biava, M. | |
Synthesis, biological evaluation, and molecular modeling of oleuropein and its semisynthetic derivatives as cyclooxygenase inhibitors | 2009 | Procopio, A; Alcaro, S; Nardi, M; Oliverio, M; Ortuso, F; Sacchetta, Paolo; Pieragostino, Damiana; Sindona, G. | |
“Synthesis, characterisation and application of a novel thiophene-based polymer” | 2005 | Cheylan, S; Fraleoni Morgera, A; Puigdollers, J; Voz, C; Alcubilla, R; Setti, L; Badenes, G | |
Synthesis, characterization and evaluation of gemfibrozil-stilbene hybrid as antioxidant agent | 2018 | Amoroso, Rosa; Leporini, Lidia; Cacciatore, Ivana; Marinelli, Lisa; Ammazzalorso, Alessandra; Bruno, Isabella; De Filippis, Barbara; Fantacuzzi, Marialuigia; Maccallini, Cristina; Menghini, Luigi; Di Stefano, Antonio; Giampietro, Letizia | |
Synthesis, characterization and optical properties of a regioregular and soluble poly [3-(10-hydroxydecyl)-2,5-thienylene] | 2003 | Lanzi, Massimiliano; Costa-Bizzarri, Paolo; Della-Casa, Carlo; FRALEONI MORGERA, Alessandro; Paganin, Luisa | |
Synthesis, characterization, and antibacterial activity of chitosan-chelated silver nanoparticles. | 2024 | Ge, J; Li, M; Fan, J; Celia, C; Xie, Y; Chang, Q; Deng, X. | |
Synthesis, characterization, and computational study of aggregates from amphiphilic calix[6]arenes. Effect of encapsulation on degradation kinetics of curcumin | 2022 | Moffa, S.; Aschi, M.; Bazzoni, M.; Cester Bonati, F.; Secchi, A.; Bruni, P.; Di Profio, P.; Fontana, A.; Pilato, S.; Siani, G. | |
Synthesis, Characterization, and DNA Binding Profile of a Macrocyclic β-Sheet Analogue of ARC Protein | 2015 | Stefanucci, Azzurra; Mosquera, Jesús; Vázquez, Eugènio; Mascareñas, José L.; Novellino, Ettore; Mollica, Adriano | |
Synthesis, crystal structure and crystal-chemistry of ferri-clinoholmquistite, Li2Mg3Fe3+2Si8O22(OH)2. | 2004 | Iezzi, Gianluca; Camara, F.; DELLA VENTURA, G.; Oberti, R.; Pedrazzi, G.; Robert, J. L. | |
Synthesis, crystal structure, and magnetic properties of a ferrimagnetic layered compound [NEt(4)][Mn(5-Cl-salen)](2)[Fe(CN)(6)] (NEt(4) equals tetraethylammonium, 5-Cl-salen equals N,N'-ethylenebis((5-chlorosalicylidene)aminato)) | 1997 | H., Miyasaka; N., Matsumoto; Re, Nazzareno; E., Gallo; C., Floriani | |
Synthesis, cytotoxicity and anti−proliferative activity against ags cells of new 3(2h)−pyridazinone derivatives endowed with a piperazinyl linker | 2021 | Alagoz, M. A.; Ozdemir, Z.; Uysal, M.; Carradori, S.; Gallorini, M.; Ricci, A.; Zara, S.; Mathew, B. | |
Synthesis, in vitro evaluation, and molecular modelling investigation of benzenesulfonimide Peroxisome Proliferator-Activated Receptors α antagonists | 2016 | Ammazzalorso, Alessandra; Carrieri, Antonio; Verginelli, Fabio; Bruno, Isabella; Carbonara, Giuseppe; D'Angelo, Alessandra; DE FILIPPIS, Barbara; Fantacuzzi, Marialuigia; Florio, Rosalba; Fracchiolla, Giuseppe; Giampietro, Letizia; Giancristofaro, Antonella; Maccallini, Cristina; Cama, Alessandro; Amoroso, Rosa | |
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents. | 2008 | Biava, M; Porretta, Gc; Poce, G; Supino, S; Manetti, F; Forli, S; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Giordani, A; Anzellotti, P; Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Anzini, M; Patrignani, Paola | |
Synthesis, magnetic properties, and incomplete double-cubane structure of Manganese(III)-metal(II) complexes [Mn(MeOH)L(OH)M(bpy)](2) (M = Zn, Cu, Ni, and Mn; H4L = 1,2-bis(2-hydroxybenzamido)benzene; bpy = 2,2 '-bipyridine) | 1998 | Y., Sunatsuki; H., Shimada; T., Matsuo; M., Nakamura; F., Kai; N., Matsumoto; Re, Nazzareno | |
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N’-bis[2-oxo-2H-benzopyran]-3-carboxamides | 2006 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Befani, O.; Turini, P.; Alcaro, S.; Ortuso, F. | |
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins | 2009 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Bizzarri, B.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Ortuso, F.; Alcaro, S. | |
Synthesis, pharmacological characterization, and docking analysis of a novel family of diarylisoxazoles as highly selective cyclooxygenase-1 (COX-1) inhibitors. | 2013 | Vitale, P; Tacconelli, Stefania; Perrone, Mg; Malerba, P; Simone, L; Scilimati, A; Lavecchia, A; Dovizio, Melania; Marcantoni, Emanuela; Bruno, Annalisa; Patrignani, Paola | |
Synthesis, Resolution, and Preliminary Evaluation of trans-2-amino-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes and Related Derivatives as Dopamine Receptors ligands | 1996 | Claudi, F; Cingolani, G. M.; DI STEFANO, Antonio; Giorgioni, G; Amenta, F; Barili, P; Ferrari, F; Giuliani, D. |
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