COSTANTE, ROBERTO
COSTANTE, ROBERTO
DIPARTIMENTO DI FARMACIA
Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice
2017-01-01 Starnowska, Joanna; Costante, Roberto; Guillemyn, Karel; Popiolek-Barczyk, Katarzyna; Chung, Nga N.; Lemieux, Carole; Keresztes, Attila; Van Duppen, Joost; Mollica, Adriano; Streicher, John; Vanden Broeck, Jozef; Schiller, Peter W.; Tourwé, Dirk; Mika, Joanna; Ballet, Steven; Przewlocka, Barbara
Antinociceptive profile of potent opioid peptide AM94, a fluorinated analogue of biphalin with non-hydrazine linker
2013-01-01 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Pinnen, Francesco Enrico; Lucente, Gino; Fidanza, Stefano; Pieretti, Stefano
Arginine- and lysine-rich peptides: Synthesis, characterization and antimicrobial activity
2018-01-01 Mollica, Adriano; Macedonio, Giorgia; Stefanucci, Azzurra; Costante, Roberto; Carradori, Simone; Cataldi, Valentina; Di Giulio, Mara; Cellini, Luigina; Silvestri, Romano; Giordano, Cesare; Scipioni, Anita; Morosetti, Stefano; Punzi, Pasqualina; Mirzaie, Sako
Biological active analogues of the opioid peptide Biphalin: mixed a/b3-peptides
2013-01-01 Mollica, Adriano; Pinnen, Francesco Enrico; Costante, Roberto; Locatelli, Marcello; Stefanucci, Azzurra; Stefano, Pieretti; Peg, Davis; Josephine, Lai; David, Rankin; Frank, Porreca; Victor J., Hruby
Cyclotides: A natural combinatorial peptide library or a bioactive sequence player?
2015-01-01 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Novellino, Ettore
Cysteine-, methionine- and seleno-cysteine-proline chimeras: Synthesis and their use in peptidomimetics design
2016-01-01 Stefanucci, Azzurra; Costante, Roberto; Macedonio, Giorgia; Dvoracsko, Szabolcs; Mollica, Adriano
Design, Synthesis and Biological Evaluation of Two Opioid Agonist and Cav2.2 Blocker Multitarget Ligands
2015-01-01 Mollica, Adriano; Costante, Roberto; Novellino, Ettore; Stefanucci, Azzurra; Pieretti, Stefano; Zador, Ferenc; Samavati, Reza; Borsodi, Anna; Benyhe, Sándor; Vetter, Irina; Lewis, Richard J.
DPP-4 inhibitors: A patent review (2012 - 2014)
2015-01-01 Costante, Roberto; Stefanucci, Azzurra; Carradori, Simone; Novellino, Ettore; Mollica, Adriano
ENANTIO-SELECTIVE SYNTHESIS OF NON-NATURAL AMINO ACIDS
2016-01-01 Mollica, Adriano; Costante, Roberto
Exploring new Probenecid-based carbonic anhydrase inhibitors: Synthesis, biological evaluation and docking studies
2015-01-01 Mollica, Adriano; Costante, Roberto; Akdemir, Atilla; Carradori, Simone; Stefanucci, Azzurra; Macedonio, Giorgia; Ceruso, Mariangela; Supuran, Claudiu T.
Exploring the biological consequences of conformational changes in aspartame models containing constrained analogues of phenylalanine
2016-01-01 Mollica, Adriano; Mirzaie, Sako; Costante, Roberto; Carradori, Simone; Macedonio, Giorgia; Stefanucci, Azzurra; Dvoracsko, Szabolcs; Novellino, Ettore
Hybrid peptides endomorphin-2/DAMGO: Design, synthesis and biological evaluation
2013-01-01 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Pinnen, Francesco Enrico; Luisi, Grazia; Stefano, Pieretti; Anna, Borsodi; Engin, Bojnik; Sándor, Benyhe
Multi-target peptides for chronic pain control: opioid agonists/omega-conotoxin analogues
2014-01-01 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra
New insight on the synthesis of neurotoxins domoic acid and kainic acid
2015-01-01 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Novellino, Ettore
Novel cyclic biphalin analogue with improved antinociceptive properties
2014-01-01 Mollica, Adriano; Carotenuto, Alfonso; Novellino, Ettore; Limatola, Antonio; Costante, Roberto; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Pieretti, Stefano; Borsodi, Anna; Samavati, Reza; Zador, Ferenc; Benyhe, Sándor; Davis, Peg; Porreca, Frank; Hruby, Victor J.
Novel Endomorphin-2 analogues: design, synthesis and biological evaluation
2012-01-01 Mollica, Adriano; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Costante, Roberto; Cacciatore, Ivana; Fornasari, Erika; S., Pieretti
Peptidi ibridi endomorfina-2/DAMGO: progettazione, sinteti e valutazione biologica
2012-01-01 Costante, Roberto; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Mollica, Adriano
Pharmacological profile of new fluorinated analogue of Biphalin with non-hydrazide linker (AM94): an update
2012-01-01 Mollica, Adriano; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Costante, Roberto; S., Pieretti
Potent Biphalin Analogs with µ/δ Mixed Opioid Activity: In Vivo and In Vitro Biological Evaluation
2013-01-01 Costante, Roberto; Stefanucci, Azzurra; Pinnen, F; Mollica, Adriano
Preparation of Constrained Unnatural Aromatic Amino Acids via Unsaturated Diketopiperazine Intermediate
2016-01-01 Mollica, Adriano; Costante, Roberto; Mirzaie, Sako; Carradori, Simone; Macedonio, Giorgia; Stefanucci, Azzurra; Novellino, Ettore
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice | 2017 | Starnowska, Joanna; Costante, Roberto; Guillemyn, Karel; Popiolek-Barczyk, Katarzyna; Chung, Nga N.; Lemieux, Carole; Keresztes, Attila; Van Duppen, Joost; Mollica, Adriano; Streicher, John; Vanden Broeck, Jozef; Schiller, Peter W.; Tourwé, Dirk; Mika, Joanna; Ballet, Steven; Przewlocka, Barbara | |
| Antinociceptive profile of potent opioid peptide AM94, a fluorinated analogue of biphalin with non-hydrazine linker | 2013 | Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Pinnen, Francesco Enrico; Lucente, Gino; Fidanza, Stefano; Pieretti, Stefano | |
| Arginine- and lysine-rich peptides: Synthesis, characterization and antimicrobial activity | 2018 | Mollica, Adriano; Macedonio, Giorgia; Stefanucci, Azzurra; Costante, Roberto; Carradori, Simone; Cataldi, Valentina; Di Giulio, Mara; Cellini, Luigina; Silvestri, Romano; Giordano, Cesare; Scipioni, Anita; Morosetti, Stefano; Punzi, Pasqualina; Mirzaie, Sako | |
| Biological active analogues of the opioid peptide Biphalin: mixed a/b3-peptides | 2013 | Mollica, Adriano; Pinnen, Francesco Enrico; Costante, Roberto; Locatelli, Marcello; Stefanucci, Azzurra; Stefano, Pieretti; Peg, Davis; Josephine, Lai; David, Rankin; Frank, Porreca; Victor J., Hruby | |
| Cyclotides: A natural combinatorial peptide library or a bioactive sequence player? | 2015 | Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Novellino, Ettore | |
| Cysteine-, methionine- and seleno-cysteine-proline chimeras: Synthesis and their use in peptidomimetics design | 2016 | Stefanucci, Azzurra; Costante, Roberto; Macedonio, Giorgia; Dvoracsko, Szabolcs; Mollica, Adriano | |
| Design, Synthesis and Biological Evaluation of Two Opioid Agonist and Cav2.2 Blocker Multitarget Ligands | 2015 | Mollica, Adriano; Costante, Roberto; Novellino, Ettore; Stefanucci, Azzurra; Pieretti, Stefano; Zador, Ferenc; Samavati, Reza; Borsodi, Anna; Benyhe, Sándor; Vetter, Irina; Lewis, Richard J. | |
| DPP-4 inhibitors: A patent review (2012 - 2014) | 2015 | Costante, Roberto; Stefanucci, Azzurra; Carradori, Simone; Novellino, Ettore; Mollica, Adriano | |
| ENANTIO-SELECTIVE SYNTHESIS OF NON-NATURAL AMINO ACIDS | 2016 | Mollica, Adriano; Costante, Roberto | |
| Exploring new Probenecid-based carbonic anhydrase inhibitors: Synthesis, biological evaluation and docking studies | 2015 | Mollica, Adriano; Costante, Roberto; Akdemir, Atilla; Carradori, Simone; Stefanucci, Azzurra; Macedonio, Giorgia; Ceruso, Mariangela; Supuran, Claudiu T. | |
| Exploring the biological consequences of conformational changes in aspartame models containing constrained analogues of phenylalanine | 2016 | Mollica, Adriano; Mirzaie, Sako; Costante, Roberto; Carradori, Simone; Macedonio, Giorgia; Stefanucci, Azzurra; Dvoracsko, Szabolcs; Novellino, Ettore | |
| Hybrid peptides endomorphin-2/DAMGO: Design, synthesis and biological evaluation | 2013 | Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Pinnen, Francesco Enrico; Luisi, Grazia; Stefano, Pieretti; Anna, Borsodi; Engin, Bojnik; Sándor, Benyhe | |
| Multi-target peptides for chronic pain control: opioid agonists/omega-conotoxin analogues | 2014 | Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra | |
| New insight on the synthesis of neurotoxins domoic acid and kainic acid | 2015 | Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Novellino, Ettore | |
| Novel cyclic biphalin analogue with improved antinociceptive properties | 2014 | Mollica, Adriano; Carotenuto, Alfonso; Novellino, Ettore; Limatola, Antonio; Costante, Roberto; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Pieretti, Stefano; Borsodi, Anna; Samavati, Reza; Zador, Ferenc; Benyhe, Sándor; Davis, Peg; Porreca, Frank; Hruby, Victor J. | |
| Novel Endomorphin-2 analogues: design, synthesis and biological evaluation | 2012 | Mollica, Adriano; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Costante, Roberto; Cacciatore, Ivana; Fornasari, Erika; S., Pieretti | |
| Peptidi ibridi endomorfina-2/DAMGO: progettazione, sinteti e valutazione biologica | 2012 | Costante, Roberto; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Mollica, Adriano | |
| Pharmacological profile of new fluorinated analogue of Biphalin with non-hydrazide linker (AM94): an update | 2012 | Mollica, Adriano; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Costante, Roberto; S., Pieretti | |
| Potent Biphalin Analogs with µ/δ Mixed Opioid Activity: In Vivo and In Vitro Biological Evaluation | 2013 | Costante, Roberto; Stefanucci, Azzurra; Pinnen, F; Mollica, Adriano | |
| Preparation of Constrained Unnatural Aromatic Amino Acids via Unsaturated Diketopiperazine Intermediate | 2016 | Mollica, Adriano; Costante, Roberto; Mirzaie, Sako; Carradori, Simone; Macedonio, Giorgia; Stefanucci, Azzurra; Novellino, Ettore |