PINNEN, Francesco Enrico

PINNEN, Francesco Enrico  

DIPARTIMENTO DI FARMACIA  

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(Acyloxy)Alkoxy Moiety as Amino Acids Protecting Group for the Synthesis of (R,R)-2,7 Diaminosuberic Acid via RCM 2012 Mollica, Adriano; Feliciani, F; Stefanucci, Azzurra; Fadeev, Ea; Pinnen, Francesco Enrico
(R)-alpha-Lipoic Acid–Gly-L-Pro-L-Glu(OMe)-OMe Codrug as Multifunctional Agent for Neurodegenerative Diseases, with Antioxidant and Neuroprotective Properties 2012 Fornasari, Erika; Cacciatore, Ivana; Cornacchia, Catia; Baldassarre, Leonardo; Pinnen, Francesco Enrico
(R)-α-Lipoyl-glycyl-L-prolyl-L-glutamyl dimethyl ester codrug as a multifunctional agent with potential neuroprotective activities 2012 Cacciatore, Ivana; Baldassarre, Leonardo; Fornasari, Erika; Cornacchia, Catia; DI STEFANO, Antonio; Sozio, Piera; Cerasa, LAURA SERAFINA; Fontana, Antonella; Fulle, Stefania; DI FILIPPO, ESTER SARA; LA ROVERE, RITA MARIA LAURA; Pinnen, Francesco Enrico
2,5-Diketopiperazines as neuroprotective agents 2012 Cornacchia, Catia; Cacciatore, Ivana; Baldassarre, Leonardo; Mollica, Adriano; Feliciani, Federica; Pinnen, Francesco Enrico
4-Amino-1,2-dithiolane-4-carboxylic acid (Adt) as Cysteine Conformationally Restricted Analogue. Synthetic Protocol for Adt Containing Peptides 2000 Morera, E; Nalli, M; Pinnen, Francesco Enrico; Rossi, D; Lucente, G.
A glutathione derivative with chelating and in vitro neuroprotective activities: synthesis, physicochemical properties, and biological evaluation. 2013 Cacciatore, Ivana; Cornacchia, C.; Fornasari, Erika; Baldassarre, L.; Pinnen, Francesco Enrico; Sozio, Piera; DI STEFANO, Antonio; Marinelli, L.; Dean, A.; Fulle, Stefania; Di Filippo, E. S.; La Rovere, R. M. L.; Patruno, Antonia; Ferrone, A.; Di Marco, V.
A new chromogenic substrate for pantetheine hydrolase and vanin proteins 2002 Dupre, Silvestro; Pinnen, Francesco Enrico; Cacciatore, Ivana; DI LEANDRO, Luana; Paolone, Tommaso; Ippoliti, Rodolfo; Pitari, Giuseppina; Malatesta, Francesco
A novel member of the GCN5-related N-acetyltransferase superfamily from Caenorhabditis elegans preferentially catalyses the N-acetylation of thialysine (S-(2-aminoethyl)-L-cysteine) 2004 ABO DALO, B; Ndjonka, D; Pinnen, Francesco Enrico; Liebau, E; Luersen, K.
A novel TRH analog containing a gamma-sultam residue replacing the pyroglutamic acid 1999 Brunetti, Luigi; DI STEFANO, Antonio; G., Lucente; Luisi, Grazia; B., Michelotto; Orlando, Giustino; Pinnen, Francesco Enrico
A Potent (R)-alpha-bis-lipoyl Derivative Containing 8-Hydroxyquinoline Scaffold: Synthesis and Biological Evaluation of Its Neuroprotective Capabilities in SH-SY5Y Human Neuroblastoma Cells 2013 Cacciatore, Ivana; Fornasari, Erika; Baldassarre, Leonardo; Cornacchia, Catia; Fulle, Stefania; DI FILIPPO, ESTER SARA; Pietrangelo, Tiziana; Pinnen, Francesco Enrico
Antinociceptive profile of potent opioid peptide AM94, a fluorinated analogue of biphalin with non-hydrazine linker 2013 Mollica, Adriano; Costante, Roberto; Stefanucci, Azzurra; Pinnen, Francesco Enrico; Lucente, Gino; Fidanza, Stefano; Pieretti, Stefano
Approaches to pseudopeptidic ergopeptines. Part 2. Consequences of the incorporation of an alfa-azaproline residue into the oxacyclolic system 1994 Pinnen, Francesco Enrico; Luisi, Grazia; Calcagni, A; Lucente, G; Gavuzzo, E; Cerrini, S.
Approaches to pseudopeptidic ergopeptines. Part 3. Consequences of the incorporation of an α-azaphenylalanine residue into the ergotamine oxa-cyclolic system 1997 Calcagni, A; Lucente, G; Luisi, Grazia; Pinnen, Francesco Enrico; Rossi, D; Gavuzzo, E.
Approaches to pseudopeptidic ergopeptines. Synthesis and molecular structure of an alfa-aza-phenylalanine-containing oxa-cyclol 1993 Pinnen, Francesco Enrico; Luisi, Grazia; Lucente, G; Gavuzzo, E; Cerrini, S.
Backbone-modified glutathione analogues 1996 A., Calcagni; S., Dupre'; G., Lucente; Luisi, Grazia; Pinnen, Francesco Enrico; D., Rossi; A., Spirito
Bicyclic peptides: Solution conformation and Ca++ binding of the heterodetic bicyclic decapeptide cyclo(Glu-Leu-Pro-Gly-Ser-Ile-Pro-Ala)-cyclo(Phe-Gly)’ 1989 Pinnen, Francesco Enrico; Zanotti, G; Lucente, G; Paolillo, L; D'Auria, G; Trivellone, E; D'Anagni, M.
Biochemical properties of new synthetic carnosine analogues containing the residue of 2,3-diaminopropionic acid: the effect of N-acetylation 2005 Cacciatore, Ivana; Cocco, Alessandra; Costa, M; Fontana, M; Lucente, G; Pecci, L; Pinnen, Francesco Enrico
Biological active analogues of the opioid peptide Biphalin: mixed a/b3-peptides 2013 Mollica, Adriano; Pinnen, Francesco Enrico; Costante, Roberto; Locatelli, Marcello; Stefanucci, Azzurra; Stefano, Pieretti; Peg, Davis; Josephine, Lai; David, Rankin; Frank, Porreca; Victor J., Hruby
cis-4-Amino-l-proline Residue As a Scaffold for the Synthesis of Cyclic and Linear Endomorphin-2 Analogues: Part 2 2012 Mollica, Adriano; Pinnen, Francesco Enrico; Stefanucci, Azzurra; Mannina, L; Sobolev, A. P.; Lucente, G; Davis, P; Lai, J; Ma, S. W.; Porreca, F; Hruby, V. J.
CNS delivery of L-Dopa by a new Hybrid Glutathione-Methionine peptidomimetic prodrug 2012 Pinnen, Francesco Enrico; Cacciatore, Ivana; Cornacchia, Catia; Mollica, Adriano; Sozio, Piera; Cerasa, LAURA SERAFINA; Iannitelli, Antonio; Fontana, Antonella; Nasuti, Cinzia; DI STEFANO, Antonio