Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors
2014-01-01 D’Ascenzio, M.; Carradori, Simone; Secci, D.; Mannina, L.; Sobolev, A. P.; De Monte, C.; Cirilli, R.; Yáñez, M.; Alcaro, S.; Ortuso, F.
CPTH6, a thiazole-derivative, induces histone hypoacetylation and apoptosis in human leukemia cells
2012-01-01 Trisciuoglio, D.; Ragazzoni, Y.; Pelosi, A.; Desideri, M.; Carradori, Simone; Gabellini, C.; Maresca, G.; Nescatelli, R.; Secci, D.; Bolasco, A.; Bizzarri, B.; Cavaliere, C.; D'Agnano, I.; Filetici, P.; Ricci Vitiani, L.; Rizzo, M. G.; Del Bufalo, D.
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
2016-01-01 De Monte, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela
Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines
2010-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Sanna, M. L.; Gallinella, B.; Cirilli, R.
Novel monoamine oxidase inhibitors: a patent review (2012-2014)
2015-01-01 Carradori, Simone; Petzer, J. P.
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives
2010-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Scaltrito, M. M.; Sisto, F.
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2010-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; Rivanera, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F.
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
2010-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Yáñez, M.; Orallo, F.
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Maccioni, E.; Cardia, M. C.; Yáñez, M.; Orallo, F.; Alcaro, S.; Ortuso, F.; Cirilli, R.; Ferretti, R.; Distinto, S.; Kirchmair, J.; Langer, T. .
Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives
2012-01-01 Carradori, Simone; Secci, D.; Bolasco, A.; De Monte, C.; Yáñez, M.
NMR methodologies in the analysis of blueberries
2014-01-01 Capitani, D.; Sobolev, A. P; Delfini, M.; Vista, S.; Antiochia, R.; Proietti, N.; Bubici, S.; Ferrante, G.; Carradori, Simone; De Salvador, F. R.; Mannina, L.
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives
2010-01-01 Chimenti, F.; Bolasco, A.; Secci, D.; Bizzarri, B.; Chimenti, P.; Granese, A.; Carradori, Simone
Selective MAO-B inhibitors: a lesson from natural products
2014-01-01 Carradori, Simone; D’Ascenzio, M.; Chimenti, P.; Secci, D.; Bolasco, A.
A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl)hydrazone
2009-01-01 Chimenti, F.; Bizzarri, B.; Maccioni, E.; Secci, D.; Bolasco, A.; Chimenti, P.; Fioravanti, R.; Granese, A.; Carradori, Simone; Tosi, F.; Ballario, P.; Vernarecci, S.; Filetici, P.
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins
2009-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Bizzarri, B.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Ortuso, F.; Alcaro, S.
Untargeted NMR-based methodologies in the study of fruits metabolites
2015-01-01 Sobolev, A. P.; Mannina, L.; Proietti, N.; Carradori, Simone; Daglia, M.; Giusti, A. M.; Antiochia, R.; Capitani, D.
Epigenetic modulation of PGC-1α activity by GCN5 inhibitors: WO2010007085
2011-01-01 Carradori, Simone; Secci, D.; Mai, A. .
Current and emerging strategies in bladder cancer
2012-01-01 Carradori, Simone; Cristini, C.; Secci, D.; Gulia, C.; Gentile, V.; Di Pierro, G. B.
New Frontiers in Selective Human MAO-B Inhibitors
2015-01-01 Carradori, Simone; Silvestri, R.
A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives
2007-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Carradori, Simone; Granese, A.; Rivanera, D.; Lilli, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors | 2014 | D’Ascenzio, M.; Carradori, Simone; Secci, D.; Mannina, L.; Sobolev, A. P.; De Monte, C.; Cirilli, R.; Yáñez, M.; Alcaro, S.; Ortuso, F. | |
| CPTH6, a thiazole-derivative, induces histone hypoacetylation and apoptosis in human leukemia cells | 2012 | Trisciuoglio, D.; Ragazzoni, Y.; Pelosi, A.; Desideri, M.; Carradori, Simone; Gabellini, C.; Maresca, G.; Nescatelli, R.; Secci, D.; Bolasco, A.; Bizzarri, B.; Cavaliere, C.; D'Agnano, I.; Filetici, P.; Ricci Vitiani, L.; Rizzo, M. G.; Del Bufalo, D. | |
| Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives | 2016 | De Monte, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela | |
| Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines | 2010 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Sanna, M. L.; Gallinella, B.; Cirilli, R. | |
| Novel monoamine oxidase inhibitors: a patent review (2012-2014) | 2015 | Carradori, Simone; Petzer, J. P. | |
| Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives | 2010 | Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Scaltrito, M. M.; Sisto, F. | |
| Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2010 | Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Granese, A.; Carradori, Simone; Rivanera, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F. | |
| Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones | 2010 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; D’Ascenzio, M.; Yáñez, M.; Orallo, F. | |
| Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 2010 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Carradori, Simone; Maccioni, E.; Cardia, M. C.; Yáñez, M.; Orallo, F.; Alcaro, S.; Ortuso, F.; Cirilli, R.; Ferretti, R.; Distinto, S.; Kirchmair, J.; Langer, T. . | |
| Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives | 2012 | Carradori, Simone; Secci, D.; Bolasco, A.; De Monte, C.; Yáñez, M. | |
| NMR methodologies in the analysis of blueberries | 2014 | Capitani, D.; Sobolev, A. P; Delfini, M.; Vista, S.; Antiochia, R.; Proietti, N.; Bubici, S.; Ferrante, G.; Carradori, Simone; De Salvador, F. R.; Mannina, L. | |
| Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives | 2010 | Chimenti, F.; Bolasco, A.; Secci, D.; Bizzarri, B.; Chimenti, P.; Granese, A.; Carradori, Simone | |
| Selective MAO-B inhibitors: a lesson from natural products | 2014 | Carradori, Simone; D’Ascenzio, M.; Chimenti, P.; Secci, D.; Bolasco, A. | |
| A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl)hydrazone | 2009 | Chimenti, F.; Bizzarri, B.; Maccioni, E.; Secci, D.; Bolasco, A.; Chimenti, P.; Fioravanti, R.; Granese, A.; Carradori, Simone; Tosi, F.; Ballario, P.; Vernarecci, S.; Filetici, P. | |
| Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins | 2009 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Bizzarri, B.; Granese, A.; Carradori, Simone; Yáñez, M.; Orallo, F.; Ortuso, F.; Alcaro, S. | |
| Untargeted NMR-based methodologies in the study of fruits metabolites | 2015 | Sobolev, A. P.; Mannina, L.; Proietti, N.; Carradori, Simone; Daglia, M.; Giusti, A. M.; Antiochia, R.; Capitani, D. | |
| Epigenetic modulation of PGC-1α activity by GCN5 inhibitors: WO2010007085 | 2011 | Carradori, Simone; Secci, D.; Mai, A. . | |
| Current and emerging strategies in bladder cancer | 2012 | Carradori, Simone; Cristini, C.; Secci, D.; Gulia, C.; Gentile, V.; Di Pierro, G. B. | |
| New Frontiers in Selective Human MAO-B Inhibitors | 2015 | Carradori, Simone; Silvestri, R. | |
| A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives | 2007 | Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Carradori, Simone; Granese, A.; Rivanera, D.; Lilli, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F. |
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Tipologia
- 1.1 Articolo in rivista46885
- 1.2 Recensione in rivista1
- 3.1 Monografia o trattato scienti...1
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Data di pubblicazione
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- 2020 - 202713655
- 2010 - 201915958
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- 1990 - 19995150
- 1980 - 19891724
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- 1967 - 19694
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