CARRADORI, SIMONE
CARRADORI, SIMONE
DIPARTIMENTO DI FARMACIA
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
2015-01-01 D’Ascenzio, M.; Chimenti, P.; Gidaro, M. C.; De Monte, C.; De Vita, D.; Granese, A.; Scipione, L.; Di Santo, R.; Costa, G.; Alcaro, S.; Yáñez, M.; Carradori, Simone
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020-01-01 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
2-Substituted Benzothiazoles as Antiproliferative Agents: Novel Insights on Structure-Activity Relationships
2020-01-01 Ammazzalorso, Alessandra; Carradori, Simone; Amoroso, Rosa; Fernández Fernández, Inmaculada
2-Substituted-4,7-dihydro-4-ethylpyrazolo[1,5-a]pyrimidin-7-ones alleviate LPS-induced inflammation by modulating cell metabolism via CD73 upon macrophage polarization
2024-01-01 Ricci, A.; Zara, S.; Carta, F.; Di Valerio, V.; Sancilio, S.; Cataldi, A.; Selleri, S.; Supuran, C. T.; Carradori, S.; Gallorini, M.
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: A fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part II. Solvophobic effects in enantiorecognition process
2017-01-01 Pierini, M.; Carradori, Simone; Menta, S.; Secci, D.; Cirilli, R.
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: A fascinatingmolecular framework to study the enantioseparation ability of theamylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part I. Structure-enantioselectivity relationships
2016-01-01 Carradori, Simone; Pierini, Marco; Menta, Sergio; Secci, Daniela; Fioravanti, Rossella; Cirilli, Roberto
3-Methylcyclohexanone thiosemicarbazone: determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes
2012-01-01 Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, S.; Pierini, M.; Secci, D.
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019-01-01 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
A chromatographic study on the exceptional chiral recognition of 2-(benzylsulfinyl)benzamide by an immobilized-type chiral stationary phase based on cellulose tris(3,5-dichlorophenylcarbamate)
2018-01-01 Carradori, Simone; Secci, Daniela; Faggi, Cristina; Cirilli, Roberto
A chromatographic study on the retention behavior of the amylose tris(3-chloro-5-methylphenylcarbamate) chiral stationary phase under aqueous conditions
2018-01-01 Cirilli, Roberto; Carradori, Simone; Casulli, Adriano; Pierini, Marco
A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases
2016-01-01 Langella, Emma; D’Ambrosio, Katia; D’Ascenzio, Melissa; Carradori, Simone; Monti, Simona M.; Supuran, Claudiu T.; De Simone, Giuseppina
A Comparative Assessment of Biological Effects and Chemical Profile of Italian Asphodeline lutea Extracts
2018-01-01 Melucci, Dora; Locatelli, Marcello; Locatelli, Clinio; Zappi, Alessandro; De Laurentiis, Francesco; Carradori, Simone; Campestre, Cristina; Leporini, Lidia; Zengin, Gokhan; Marie Nancy Picot, Carene; Menghini, Luigi; Fawzi Mahomoodally, Mohamad
A Comprehensive Overview of Colon Cancer- A Grim Reaper of the 21st Century
2021-01-01 Kumar, R.; Harilal, S.; Carradori, S.; Mathew, B.
A multi-methodological approach in the study of Italian PDO “Cornetto di Pontecorvo
2018-01-01 Sobolev, Anatoly P.; Mannina, Luisa; Capitani, Donatella; Sanzò, Gabriella; Ingallina, Cinzia; Botta, Bruno; Fornarini, Simonetta; Elisa Crestoni, Maria; Chiavarino, Barbara; Carradori, Simone; Locatelli, Marcello; Maria Giusti, Anna; Simonetti, Giovanna; Vinci, Giuliana; Preti, Raffaella; Toniolo, Chiara; Reverberi, Massimo; Scarpari, Marzia; Parroni, Alessia; Abete, Lorena; Natella, Fausta; Sotto., Antonella Di
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023-01-01 Berrino, Emanuela; Carradori, Simone; Carta, Fabrizio; Melfi, Francesco; Gallorini, Marialucia; Poli, Giulio; Tuccinardi, Tiziano; Fernández-Bolaños, José G; López, Óscar; Petzer, Jacobus P; Petzer, Anél; Guglielmi, Paolo; Secci, Daniela; Supuran, Claudiu T
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes
2021-01-01 Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G.
A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives
2007-01-01 Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Carradori, Simone; Granese, A.; Rivanera, D.; Lilli, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F.
A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl)hydrazone
2009-01-01 Chimenti, F.; Bizzarri, B.; Maccioni, E.; Secci, D.; Bolasco, A.; Chimenti, P.; Fioravanti, R.; Granese, A.; Carradori, Simone; Tosi, F.; Ballario, P.; Vernarecci, S.; Filetici, P.
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016-01-01 Carradori, Simone; Secci, Daniela; Monte, Celeste De; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P.; Codispoti, Rossella; Cosmi, Federica De; Guglielmi, Paolo; Supuran, Claudiu T.
A novel life for antitumor combretastatins: Recent developments of hybrids, prodrugs, combination therapies, and antibody-drug conjugates
2024-01-01 Fantacuzzi, Marialuigia; Carradori, Simone; Giampietro, Letizia; Maccallini, Cristina; De Filippis, Barbara; Amoroso, Rosa; Ammazzalorso, Alessandra
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies | 2015 | D’Ascenzio, M.; Chimenti, P.; Gidaro, M. C.; De Monte, C.; De Vita, D.; Granese, A.; Scipione, L.; Di Santo, R.; Costa, G.; Alcaro, S.; Yáñez, M.; Carradori, Simone | |
| 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
| 2-Substituted Benzothiazoles as Antiproliferative Agents: Novel Insights on Structure-Activity Relationships | 2020 | Ammazzalorso, Alessandra; Carradori, Simone; Amoroso, Rosa; Fernández Fernández, Inmaculada | |
| 2-Substituted-4,7-dihydro-4-ethylpyrazolo[1,5-a]pyrimidin-7-ones alleviate LPS-induced inflammation by modulating cell metabolism via CD73 upon macrophage polarization | 2024 | Ricci, A.; Zara, S.; Carta, F.; Di Valerio, V.; Sancilio, S.; Cataldi, A.; Selleri, S.; Supuran, C. T.; Carradori, S.; Gallorini, M. | |
| 3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: A fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part II. Solvophobic effects in enantiorecognition process | 2017 | Pierini, M.; Carradori, Simone; Menta, S.; Secci, D.; Cirilli, R. | |
| 3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: A fascinatingmolecular framework to study the enantioseparation ability of theamylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part I. Structure-enantioselectivity relationships | 2016 | Carradori, Simone; Pierini, Marco; Menta, Sergio; Secci, Daniela; Fioravanti, Rossella; Cirilli, Roberto | |
| 3-Methylcyclohexanone thiosemicarbazone: determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes | 2012 | Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, S.; Pierini, M.; Secci, D. | |
| 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco | |
| A chromatographic study on the exceptional chiral recognition of 2-(benzylsulfinyl)benzamide by an immobilized-type chiral stationary phase based on cellulose tris(3,5-dichlorophenylcarbamate) | 2018 | Carradori, Simone; Secci, Daniela; Faggi, Cristina; Cirilli, Roberto | |
| A chromatographic study on the retention behavior of the amylose tris(3-chloro-5-methylphenylcarbamate) chiral stationary phase under aqueous conditions | 2018 | Cirilli, Roberto; Carradori, Simone; Casulli, Adriano; Pierini, Marco | |
| A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases | 2016 | Langella, Emma; D’Ambrosio, Katia; D’Ascenzio, Melissa; Carradori, Simone; Monti, Simona M.; Supuran, Claudiu T.; De Simone, Giuseppina | |
| A Comparative Assessment of Biological Effects and Chemical Profile of Italian Asphodeline lutea Extracts | 2018 | Melucci, Dora; Locatelli, Marcello; Locatelli, Clinio; Zappi, Alessandro; De Laurentiis, Francesco; Carradori, Simone; Campestre, Cristina; Leporini, Lidia; Zengin, Gokhan; Marie Nancy Picot, Carene; Menghini, Luigi; Fawzi Mahomoodally, Mohamad | |
| A Comprehensive Overview of Colon Cancer- A Grim Reaper of the 21st Century | 2021 | Kumar, R.; Harilal, S.; Carradori, S.; Mathew, B. | |
| A multi-methodological approach in the study of Italian PDO “Cornetto di Pontecorvo | 2018 | Sobolev, Anatoly P.; Mannina, Luisa; Capitani, Donatella; Sanzò, Gabriella; Ingallina, Cinzia; Botta, Bruno; Fornarini, Simonetta; Elisa Crestoni, Maria; Chiavarino, Barbara; Carradori, Simone; Locatelli, Marcello; Maria Giusti, Anna; Simonetti, Giovanna; Vinci, Giuliana; Preti, Raffaella; Toniolo, Chiara; Reverberi, Massimo; Scarpari, Marzia; Parroni, Alessia; Abete, Lorena; Natella, Fausta; Sotto., Antonella Di | |
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Berrino, Emanuela; Carradori, Simone; Carta, Fabrizio; Melfi, Francesco; Gallorini, Marialucia; Poli, Giulio; Tuccinardi, Tiziano; Fernández-Bolaños, José G; López, Óscar; Petzer, Jacobus P; Petzer, Anél; Guglielmi, Paolo; Secci, Daniela; Supuran, Claudiu T | |
| A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes | 2021 | Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. | |
| A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives | 2007 | Chimenti, F.; Bizzarri, B.; Bolasco, A.; Secci, D.; Chimenti, P.; Carradori, Simone; Granese, A.; Rivanera, D.; Lilli, D.; Zicari, A.; Scaltrito, M. M.; Sisto, F. | |
| A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl)hydrazone | 2009 | Chimenti, F.; Bizzarri, B.; Maccioni, E.; Secci, D.; Bolasco, A.; Chimenti, P.; Fioravanti, R.; Granese, A.; Carradori, Simone; Tosi, F.; Ballario, P.; Vernarecci, S.; Filetici, P. | |
| A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms | 2016 | Carradori, Simone; Secci, Daniela; Monte, Celeste De; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P.; Codispoti, Rossella; Cosmi, Federica De; Guglielmi, Paolo; Supuran, Claudiu T. | |
| A novel life for antitumor combretastatins: Recent developments of hybrids, prodrugs, combination therapies, and antibody-drug conjugates | 2024 | Fantacuzzi, Marialuigia; Carradori, Simone; Giampietro, Letizia; Maccallini, Cristina; De Filippis, Barbara; Amoroso, Rosa; Ammazzalorso, Alessandra |