DI STEFANO, Antonio
DI STEFANO, Antonio
DIPARTIMENTO DI FARMACIA
(R)-α-Lipoyl-Gly-L-Pro-L-Glu dimethyl ester as dual acting agent for the treatment of Alzheimer's disease
2017-01-01 Marinelli, Lisa; Fornasari, Erika; Di Stefano, Antonio; Turkez, Hasan; Arslan, Mehmet Enes; Eusepi, Piera; Ciulla, Michele; Cacciatore, Ivana
(R)-α-Lipoyl-glycyl-L-prolyl-L-glutamyl dimethyl ester codrug as a multifunctional agent with potential neuroprotective activities
2012-01-01 Cacciatore, Ivana; Baldassarre, Leonardo; Fornasari, Erika; Cornacchia, Catia; DI STEFANO, Antonio; Sozio, Piera; Cerasa, LAURA SERAFINA; Fontana, Antonella; Fulle, Stefania; DI FILIPPO, ESTER SARA; LA ROVERE, RITA MARIA LAURA; Pinnen, Francesco Enrico
A glutathione derivative with chelating and in vitro neuroprotective activities: synthesis, physicochemical properties, and biological evaluation.
2013-01-01 Cacciatore, Ivana; Cornacchia, C.; Fornasari, Erika; Baldassarre, L.; Pinnen, Francesco Enrico; Sozio, Piera; DI STEFANO, Antonio; Marinelli, L.; Dean, A.; Fulle, Stefania; Di Filippo, E. S.; La Rovere, R. M. L.; Patruno, Antonia; Ferrone, A.; Di Marco, V.
A new lipophilic molecular combination codrug-1 exerts neuroprotective activity in beta amyloid (1-40) infused Alzheimer’s disease rat model
2011-01-01 Zara, Susi; DI STEFANO, Antonio; M., Rapino; D., Bosco; DI GIACOMO, Viviana; Sozio, Piera; A., Abbadessa; Cataldi, Amelia
A Novel Prodrug of a nNOS Inhibitor with Improved Pharmacokinetic Potential
2020-01-01 Maccallini, C.; Marinelli, L.; Indorf, P.; Cacciatore, I.; Fantacuzzi, M.; Clement, B.; Di Stefano, A.; Amoroso, R.
A novel TRH analog containing a gamma-sultam residue replacing the pyroglutamic acid
1999-01-01 Brunetti, Luigi; DI STEFANO, Antonio; G., Lucente; Luisi, Grazia; B., Michelotto; Orlando, Giustino; Pinnen, Francesco Enrico
Activity of N-(2-phenylethyl)-N-n-propyl-(2-(3-hydroxyphenyl)ethylamine derivates as dopamine receptor ligands
1994-01-01 Claudi, F; Cardellini, M; DI STEFANO, Antonio; Giorgioni, G; Cantalamessa, F; Ren, F; Balduini, W.
Advances in Parkinson’s disease drugs
2021-01-01 Di Stefano, A.; Marinelli, L.
Advances in prodrug design for Parkinson's disease
2018-01-01 Cacciatore, Ivana; Ciulla, Michele; Marinelli, Lisa; Eusepi, Piera; Di Stefano, Antonio
Analytical Methods to Best Detect Fluorescent Probe Loading Nanoparticles in Biological Samples
2015-01-01 Primavera, Rosita; Francesco, Martina Di; Paolino, Donatella; Carafa, Maria; Cristiano, Maria Chiara; Celia, Christian; Fresta, Massimo; DI STEFANO, Antonio; Locatelli, Marcello; DI MARZIO, Luisa
Anticancer effects of novel NSAIDs derivatives on cultured human glioblastoma cells
2021-01-01 Ozdemir, O; Marinelli, L; Cacciatore, I; Ciulla, M; Emsen, B; Di Stefano, A; Mardinoglu, A; Turkez, H
Antifungal Activity of Novel Formulations Based on Terpenoid Prodrugs against C. albicans in a Mouse Model
2021-01-01 Menon, S.; Liang, X.; Vartak, R.; Patel, K.; Di Stefano, A.; Cacciatore, I.; Marinelli, L.; Billack, B.
Antiparkinson Prodrugs
2008-01-01 DI STEFANO, Antonio; Sozio, Piera; Cerasa, LAURA SERAFINA
Au nanoparticles functionalized by newly synthetised antiparkinson prodrugs
2011-01-01 E., Di Meo; S., Laserra; A., Abbadessa; Angelini, Guido; DI STEFANO, Antonio; Fontana, Antonella
Benzimidazole, benzoxazole and benzothiazole derivatives as 5HT2B receptor ligands. Synthesis and preliminary pharmacological evaluation
2005-01-01 Giorgioni, G.; Accorroni, B.; DI STEFANO, Antonio; Marucci, G.; Siniscalchi, A.; Claudi, F.
Binding and preliminary evaluation of 5-hydroxy- and 10-hydroxy-2,3, 12,12a-tetrahydro-1H-[1]benzoxepino[2,3,4-ij]isoquinolines as dopamine receptor ligands.
2000-01-01 Claudi, F; DI STEFANO, Antonio; Napolitani, F; Cingolani, Gm; Giorgioni, G; Fontenla, Ja; Montenegro, Gy; Rivas, Me; Rosa, E; Michelotto, B; Orlando, Giustino; Brunetti, Luigi
Biodegradable microspheres loaded with an antiparkinson prodrug: an in vivo pharmacokinetic study
2011-01-01 D'Aurizio, Eleonora; Sozio, Piera; Cerasa, LAURA SERAFINA; Vacca, Michele; Brunetti, Luigi; Orlando, Giustino; Chiavaroli, Annalisa; Kok, R.; Hennink, W. E.; DI STEFANO, Antonio
Boron-based hybrids as novel scaffolds for the development of drugs with neuroprotective properties
2021-01-01 Cacciatore, I.; Turkez, H.; Di Rienzo, A.; Ciulla, M.; Mardinoglu, A.; Di Stefano, A.
Carvacrol and its derivatives as antibacterial agents
2018-01-01 Marinelli, Lisa; Di Stefano, Antonio; Cacciatore, Ivana
Carvacrol codrugs: A new approach in the antimicrobial plan
2015-01-01 Cacciatore, Ivana; DI GIULIO, Mara; Fornasari, Erika; DI STEFANO, Antonio; Cerasa, LAURA SERAFINA; Marinelli, Lisa; Turkez, Hasan; DI CAMPLI, Emanuela; DI BARTOLOMEO, Soraya; Robuffo, Iole; Cellini, Luigina
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(R)-α-Lipoyl-Gly-L-Pro-L-Glu dimethyl ester as dual acting agent for the treatment of Alzheimer's disease | 2017 | Marinelli, Lisa; Fornasari, Erika; Di Stefano, Antonio; Turkez, Hasan; Arslan, Mehmet Enes; Eusepi, Piera; Ciulla, Michele; Cacciatore, Ivana | |
(R)-α-Lipoyl-glycyl-L-prolyl-L-glutamyl dimethyl ester codrug as a multifunctional agent with potential neuroprotective activities | 2012 | Cacciatore, Ivana; Baldassarre, Leonardo; Fornasari, Erika; Cornacchia, Catia; DI STEFANO, Antonio; Sozio, Piera; Cerasa, LAURA SERAFINA; Fontana, Antonella; Fulle, Stefania; DI FILIPPO, ESTER SARA; LA ROVERE, RITA MARIA LAURA; Pinnen, Francesco Enrico | |
A glutathione derivative with chelating and in vitro neuroprotective activities: synthesis, physicochemical properties, and biological evaluation. | 2013 | Cacciatore, Ivana; Cornacchia, C.; Fornasari, Erika; Baldassarre, L.; Pinnen, Francesco Enrico; Sozio, Piera; DI STEFANO, Antonio; Marinelli, L.; Dean, A.; Fulle, Stefania; Di Filippo, E. S.; La Rovere, R. M. L.; Patruno, Antonia; Ferrone, A.; Di Marco, V. | |
A new lipophilic molecular combination codrug-1 exerts neuroprotective activity in beta amyloid (1-40) infused Alzheimer’s disease rat model | 2011 | Zara, Susi; DI STEFANO, Antonio; M., Rapino; D., Bosco; DI GIACOMO, Viviana; Sozio, Piera; A., Abbadessa; Cataldi, Amelia | |
A Novel Prodrug of a nNOS Inhibitor with Improved Pharmacokinetic Potential | 2020 | Maccallini, C.; Marinelli, L.; Indorf, P.; Cacciatore, I.; Fantacuzzi, M.; Clement, B.; Di Stefano, A.; Amoroso, R. | |
A novel TRH analog containing a gamma-sultam residue replacing the pyroglutamic acid | 1999 | Brunetti, Luigi; DI STEFANO, Antonio; G., Lucente; Luisi, Grazia; B., Michelotto; Orlando, Giustino; Pinnen, Francesco Enrico | |
Activity of N-(2-phenylethyl)-N-n-propyl-(2-(3-hydroxyphenyl)ethylamine derivates as dopamine receptor ligands | 1994 | Claudi, F; Cardellini, M; DI STEFANO, Antonio; Giorgioni, G; Cantalamessa, F; Ren, F; Balduini, W. | |
Advances in Parkinson’s disease drugs | 2021 | Di Stefano, A.; Marinelli, L. | |
Advances in prodrug design for Parkinson's disease | 2018 | Cacciatore, Ivana; Ciulla, Michele; Marinelli, Lisa; Eusepi, Piera; Di Stefano, Antonio | |
Analytical Methods to Best Detect Fluorescent Probe Loading Nanoparticles in Biological Samples | 2015 | Primavera, Rosita; Francesco, Martina Di; Paolino, Donatella; Carafa, Maria; Cristiano, Maria Chiara; Celia, Christian; Fresta, Massimo; DI STEFANO, Antonio; Locatelli, Marcello; DI MARZIO, Luisa | |
Anticancer effects of novel NSAIDs derivatives on cultured human glioblastoma cells | 2021 | Ozdemir, O; Marinelli, L; Cacciatore, I; Ciulla, M; Emsen, B; Di Stefano, A; Mardinoglu, A; Turkez, H | |
Antifungal Activity of Novel Formulations Based on Terpenoid Prodrugs against C. albicans in a Mouse Model | 2021 | Menon, S.; Liang, X.; Vartak, R.; Patel, K.; Di Stefano, A.; Cacciatore, I.; Marinelli, L.; Billack, B. | |
Antiparkinson Prodrugs | 2008 | DI STEFANO, Antonio; Sozio, Piera; Cerasa, LAURA SERAFINA | |
Au nanoparticles functionalized by newly synthetised antiparkinson prodrugs | 2011 | E., Di Meo; S., Laserra; A., Abbadessa; Angelini, Guido; DI STEFANO, Antonio; Fontana, Antonella | |
Benzimidazole, benzoxazole and benzothiazole derivatives as 5HT2B receptor ligands. Synthesis and preliminary pharmacological evaluation | 2005 | Giorgioni, G.; Accorroni, B.; DI STEFANO, Antonio; Marucci, G.; Siniscalchi, A.; Claudi, F. | |
Binding and preliminary evaluation of 5-hydroxy- and 10-hydroxy-2,3, 12,12a-tetrahydro-1H-[1]benzoxepino[2,3,4-ij]isoquinolines as dopamine receptor ligands. | 2000 | Claudi, F; DI STEFANO, Antonio; Napolitani, F; Cingolani, Gm; Giorgioni, G; Fontenla, Ja; Montenegro, Gy; Rivas, Me; Rosa, E; Michelotto, B; Orlando, Giustino; Brunetti, Luigi | |
Biodegradable microspheres loaded with an antiparkinson prodrug: an in vivo pharmacokinetic study | 2011 | D'Aurizio, Eleonora; Sozio, Piera; Cerasa, LAURA SERAFINA; Vacca, Michele; Brunetti, Luigi; Orlando, Giustino; Chiavaroli, Annalisa; Kok, R.; Hennink, W. E.; DI STEFANO, Antonio | |
Boron-based hybrids as novel scaffolds for the development of drugs with neuroprotective properties | 2021 | Cacciatore, I.; Turkez, H.; Di Rienzo, A.; Ciulla, M.; Mardinoglu, A.; Di Stefano, A. | |
Carvacrol and its derivatives as antibacterial agents | 2018 | Marinelli, Lisa; Di Stefano, Antonio; Cacciatore, Ivana | |
Carvacrol codrugs: A new approach in the antimicrobial plan | 2015 | Cacciatore, Ivana; DI GIULIO, Mara; Fornasari, Erika; DI STEFANO, Antonio; Cerasa, LAURA SERAFINA; Marinelli, Lisa; Turkez, Hasan; DI CAMPLI, Emanuela; DI BARTOLOMEO, Soraya; Robuffo, Iole; Cellini, Luigina |